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ALL ABOUT DRUGS BY DR ANTHONY · 1w ago

Award for me, 100 Most Impactful Health care Leaders, Global listing

At award function for my award “100 Most Impactful Health care Leaders Global listing”, conferred on me at Taj lands end, Mumbai, India on 14 Feb 2014 by World Health Wellness congress and a...
ALL ABOUT DRUGS BY DR ANTHONY · 1W ago

tert-butyl(3aR,6aS)-5-oxohexahydrocyclopenta[c]pyrrole-2(1H)-carboxylate

  tert-butyl(3aR,6aS)-5-oxohexahydrocyclopenta[c]pyrrole-2(1H)-carboxylate tert-Butyl (3aR,6aS)-5-Oxohexahydrocyclopenta[c]pyrrole-2(1H)-carboxylate (1) pure compound 1 (1.051 kg, 67%) as a ...
ALL ABOUT DRUGS BY DR ANTHONY · 1W ago

(3R)-4-[2-chloro-6-[[(R)-methylsulfinyl]methyl]pyrimidin-4-yl]-3-methyl-morpholine

  (3R)-4-[2-chloro-6-[[(R)-methylsulfinyl]methyl]pyrimidin-4-yl]-3-methyl-morpholine Synthesis of (3R)-4-[2-chloro-6-[[(R)-methylsulfinyl]methyl]pyrimidin-4-yl]-3-methyl-morpholine (10) off-...
ALL ABOUT DRUGS BY DR ANTHONY · 1W ago

(±)-trans-ethyl 2-(3,4-difluorophenyl)Cyclopropanecarboxylate

(±)-trans-ethyl 2-(3,4-difluorophenyl)Cyclopropanecarboxylate C12H12F2O2 GC-MS (EI) m/z: [M]+ calc. for C12H12F2O2 + : 226.08; found: 226.08. δH (400 MHz, CDCl3): 1.25 (1H, ddd, 3 J 8.4 Hz, ...
ALL ABOUT DRUGS BY DR ANTHONY · 2W ago

tert-Butyl 3a,4,7,7a-Tetrahydro-1H-isoindole-2(3H)-carboxylate

  tert-Butyl 3a,4,7,7a-Tetrahydro-1H-isoindole-2(3H)-carboxylate tert-Butyl 3a,4,7,7a-Tetrahydro-1H-isoindole-2(3H)-carboxylate   as a brown oil. % Purity: 93.72% (GC); 1H NMR (CDCl3, 400 MH...
ALL ABOUT DRUGS BY DR ANTHONY · 3W ago

2,2′-(1-(tert-Butoxycarbonyl)pyrrolidine-3,4-diyl)diacetic Acid

  2,2′-(1-(tert-Butoxycarbonyl)pyrrolidine-3,4-diyl)diacetic Acid 2,2′-(1-(tert-Butoxycarbonyl)pyrrolidine-3,4-diyl)diacetic Acid  as a white solid. Mp: 162–163 °C, % purity: 94.09% (HPLC); ...
ALL ABOUT DRUGS BY DR ANTHONY · 3W ago

Dimethyl 4,4′-(Benzylazanediyl)(2E,2′E)-bis(but-2-enoate)

Dimethyl 4,4′-(Benzylazanediyl)(2E,2′E)-bis(but-2-enoate) IR (CHCl3): ν = 758, 1215, 1278, 1437, 1660, 1720, 2806, 2953, 3020, 3421 cm–1;   13C NMR (CDCl3, 100 MHz) δ: 51.53, 53.42, 58.37, 1...
ALL ABOUT DRUGS BY DR ANTHONY · 4W ago

1-Bromo-4-fluoro-2-((2-iodobenzyl)oxy)benzene

1-Bromo-4-fluoro-2-((2-iodobenzyl)oxy)benzene CAS 1161931-51-6 Mp 89.8–92.3 °C. IR (neat, ATR): 3072 (w), 1482 (s), 1451 (s), 1294 (s), 1294 (s) cm–1. 1H NMR (399 MHz, DMSO-d6) δ 5.12 (s, 2H...
ALL ABOUT DRUGS BY DR ANTHONY · 4W ago

One-Pot Reductive Cyclisations of Nitroanilines to Imidazoles

Hana and co-workers ( Synlett 2010, 18, 2759−2764) from Genentech have developed a single-step procedure for conversion of 2-nitro aromatic amines to benzimidazoles. Addition of ammonium chl...
ALL ABOUT DRUGS BY DR ANTHONY · 4W ago

Telcagepant Revisited

Telcagepant, MK-0974 Molecular FormulaC26H27F5N6O3 Average mass566.523 Da 1-piperidinecarboxamide, N-[(3R,6S)-6-(2,3-difluorophenyl)hexahydro-2-oxo-1-(2,2,2-trifluoroethyl)-1H-azepin-3-yl]-4...